Our Selective Inhibitors for Histone Methyltransferases:

UNC0638: G9a/GLP (PMID: 21743462)

UNC0642: G9a/GLP (in vivo probe) (PMID: 24102134)

MS012: GLP (PMID: 28662962)

UNC1999: EZH2/EZH1 (Orally bioavailable) (PMID: 23614352)

MS2177 (UNC0379) & MS453 (Covalent inhibitor): SETD8 (PMID: 27804297)

SGC707: PRMT3 (PMID: 25728001)

MS023: Type I PRMTs (PMID: 26598975)

MS049: Dual CARM1 and PRMT6 (PMID: 27584694)

HUK1-121: CARM1 (PMID: 28042453)