Our Selective Inhibitors for Histone Methyltransferases:
UNC0638: G9a/GLP (PMID: 21743462)
UNC0642: G9a/GLP (in vivo probe) (PMID: 24102134)
MS012: GLP (Glucagon-like peptide ) (PMID: 28662962)
UNC1999: EZH2/EZH1 (Orally bioavailable) (PMID: 23614352)
MS2177 (UNC0379) & MS453 (Covalent inhibitor): SETD8 (PMID: 27804297)
SGC707: PRMT3 (PMID: 25728001)
MS023: Type I PRMTs (PMID: 26598975)
MS049: Dual CARM1 and PRMT6 (PMID: 27584694)